DATASHEET
Formulation
Powder
Storage:
Stable for 2 years after receipt when stored at -20°C.
Product Information:
CAS Number: 315-72-0
Molecular formula: C23H29N3O
Molecular weight: 363.5
Purity: >98% (HPLC)
Appearance: Yellow powder.
Solubility: Soluble in chloroform.
InChiKey: YNZFUWZUGRBMHL-UHFFFAOYSA-N
SMILES: OCCN1CCN(CCCN2C3=CC=CC=C3C=CC3=CC=CC=C23)CC1
SMILES: OCCN1CCN(CCCN2C3=CC=CC=C3C=CC3=C2C=CC=C3)CC1
Description:
Tricyclic antidepressant and anxiolytic compound. Acts as a high affinity sigma receptor agonist, primarily at the sigma1 subtype, but also at the sigma2 subtype with somewhat lower affinity. Shows a low to moderate antagonistic affinity for the D2, 5-HT2, H1, H2, and muscarinic acetylcholine receptors. H1 and H2 receptor antagonism account for its antihistamine effects, and muscarinic acetylcholine receptor antagonism is responsible for its anticholinergic properties.