bs-82025C

DATASHEET

Formulation yellow solid

Storage: RT

Product Information:

Potent (EC50 = 1.3nM) and selective Leukotriene D4 antagonist(LTD4)1 displaying inverse agonist activity2, Blocks binding of LTD4 to human (Ki = 0.22 nM) and guinea pig (Ki = 2.1 nM) lung membranes. Selective for the CysLT1 receptor. Multidrug resistance protein 1 (MRP1) inhibitor.3

Description:

CAS Number: 115104-28-4; Chemical Name: 5-(3-(2-(7-Chloroquinolin-2-yl)ethenyl)phenyl)-8-dimethylcarbamyl-4,6-dithiaoctanoic acid; Molecular weight: 515.09; Formula: C26H27ClN2O3S2; Solubility: DMSO (50 mg/ml); Physical Properties: Yellow solid; Purity: 95% by TLC [10% methanol in methylene chloride; Rf = 0.34] NMR conforms

Size: 5mg, 25mg

Applications: Life Science(N/A)

For research use only. Not intended for diagnostic or therapeutic use.