bs-82058C

DATASHEET

Formulation Off-White solid

Storage: RT

Product Information:

Vanilloid receptor I (TRPV1) antagonist, IC50 = 35 nM for capsaicin-induced and 6 nM for acid-induced TRPV1 activation. Displays analgesic activity in rat models of neuropathic pain. Orally active and cell permeable.

Description:

CAS Number: 393514-24-4; Chemical Name: 4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide; Molecular weight: 372.9; Formula: C20H25ClN4O; Solubility: DMSO (25 mg/ml) Ethanol (15 mg/ml); Physical Properties: Off-white solid; Purity: 98% by TLC [ 2% CH3OH in CH2Cl2; Rf = 0.25] NMR Conforms

Size: 10mg, 50mg

Applications: Life Science(N/A)

For research use only. Not intended for diagnostic or therapeutic use.