DATASHEET
Formulation
White Solid
Storage:
-20°C
Product Information:
Potent and selective phosphodiesterase (PDE3) inhibitor, IC50=36 nM).1 Inhibits platelet production by disrupting megakaryocyte maturation2 via a mechanism which is independent of PDE3 inhibition3. Clinically useful agent for conditions requiring platelet lowering therapy.4,5
Description:
CAS Number: 58579-51-4; Chemical Name: 6,7-dichloro-1,5-dihydroimidazo[2,1 –b]quinazolin-2(3H)-one hydrochloride; Molecular weight: 292.55; Formula: C10H7Cl2N3O HCl; Solubility: DMSO (2.5 mg/ml); Physical Properties: White solid; Purity: 98% by HPLC, NMR (Conforms)