bs-82216C
[Life Science]
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support@biossusa.com
800.501.7654 [DOMESTIC]
+1.781.569.5821 [INTERNATIONAL]
DATASHEET
Formulation White solid
Storage: -20°C
Product Information:
Potent and selective antagonist of the platelet activating factor (PAF) receptor (Ki = 16.3 nM)1. Displays an activity profile which includes antiinflamatory, antiangiogenesis and anticancer activity2. Along with leukotriene antagonists, cooperatively provides a robust anti-inflammatory effect regulating PMNL migration and edema formation3. Displays analgesic effects in animal models of neuropathic pain4. Active in vivo.
Description:
CAS Number: 105219-56-5<br></br>Chemical Name: 4-[3-[4[(2-Chlorophenyl)-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a]diazepin-2-yl]-1-oxopropyl]morpholine<br></br>Molecular weight: 455.96<br></br>Formula: C22H22ClN5O2S<br></br>Solubility: DMSO (>50 mg/ml) Ethanol (25 mg/ml)<br></br>Physical Properties: White solid<br></br>Purity: 98% by TLC, NMR (Conforms)
Size: 1mg, 5mg
Applications: Life Science
For research use only. Not intended for diagnostic or therapeutic use.