bs-82312C [Life Science]
GAC Inhibitor 968
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Formulation Off-White solid

Storage: RT

Product Information:

Allosteric inhibitor of glutaminase C (GAC).1 Inhibition of GAC blocks oncogenic transformation induced by Rho GTPases in fibroblasts and B lymphoma cells with no effect on normal cells.2 Inhibits liver-type glutaminase GLS2 and suppresses breast tumor growth in vivo.3,4 Reverses acquired erlotinib resistance in non-small cell lung cancer.5

Description:

CAS Number: 311795-38-7; Chemical Name: 5-(3-bromo-4-(dimethylamino)phenyl)-2,2-dimethyl-2,3,5,6-tetrahydrobenzo[a]-phenanthridin-4(1H)-; Molecular weight: 475.42; Formula: C27H27BrN2O; Solubility: DMSO (11 mg/ml) Ethanol (1 mg/ml); Physical Properties: Off-white solid; Purity: 98% by TLC NMR (Conforms)

Size: 5mg, 25mg

Applications: Life Science(N/A)

For research use only. Not intended for diagnostic or therapeutic use.