DATASHEET
Formulation
solid
Storage:
-20°C
Product Information:
GDC-0941 is a potent and selective inhibitor of class I phosphatidylinositol-3-kinases (PI3K) with significant antitumor activity – IC50’s: PI3Kα = 3nM, PI3Kβ = 33 nM, PI3Kδ = 3 nM, PI3Kγ = 75 nM.1,2 GDC-0941 is the chemical probe of choice for the pan-inhibition of class I PI3K’s.3 Currently in clinical trials.4
Description:
CAS Number: 957054-30-7; Chemical Name:; Molecular weight: 513.64; Formula: C23H27N7O3S2; Solubility: DMSO (50 mg/ml); Physical Properties: solid; Purity: 98% by HPLC NMR (Conforms)