DATASHEET
Formulation
Off-white solid
Storage:
-20°C
Product Information:
H-89 is a commonly used inhibitor of protein kinase A (PKA IC50 = 140 nM). Inhibits a variety of other kinases including S6K1 (IC50 = 80 nM), MSK1 (120 nM), ROCK II (270 nM), PKBα (2.6 µM), PKD, PRK2, RSK1 and 2, SGK, AMPK, CHK1 and MAPKAP-K1b (2.8 µM).1,2
Description:
CAS Number: 127243-85-0<br></br>Chemical Name: N-[2-[[3-(4-Bromophenyl)-2-propen-1-yl]amino]ethyl]-5-isoquinolinesulfonamide dihydrochloride<br></br>Molecular weight: 519.28<br></br>Formula: C20H20BrN3O2S·2HCl <br></br>Solubility: DMSO (50 mg/ml) Water (10 mg/ml)<br></br>Physical Properties: Off-white solid<br></br>Purity: 98% by TLC NMR (Conforms)