DATASHEET
Formulation
White Solid
Storage:
RT
Product Information:
A semi-synthetic ergoline derivative which acts as a partial dopamine D2 agonist and 5HT2B/2C receptor antagonist. Displays antiparkinsonian effects in MPTP-treated cynomolgus monkeys1. Partial agonist at recruitment of -arrestin2 to the D2 receptor2. Ameliorates monocrotaline-induced pulmonary hypertension in rats3.
Description:
CAS Number: 37686-84-3; Chemical Name: S(+)-N,N-Diethyl-N′([8α]-6-methylergolin-8-yl)urea; Molecular weight: 340.47; Formula: C20H28N4O; Solubility: DMSO or Ethanol; Physical Properties: White solid; Purity: 98% by TLC, NMR (conforms)