DATASHEET
Formulation
White solid
Storage:
RT
Product Information:
Improves obesity-related metabolic dysfunction in mouse models.1 Increases thermogenesis and weight loss, decreases steatosis and improves insulin sensitivity. Inhibits TANK-binding kinase 1 (TBK1) and IKK (IC50=1.2 M).2 Clinically useful in the treatment of aphthus ulcers.3 Inhibits prostate tumor metastasis by targeting IKK/TBK1/NFB signaling.4
Description:
CAS Number: 68302-57-8<br></br>Chemical Name: TBK1 inhibitor / Antidiabetic<br></br>Molecular Weight: 298.29<br></br>Formula: C16H14N2O4<br></br>Solubility: DMSO (60 mg/ml)<br></br>Physical Properties: White solid<br></br>Purity: 98%, NMR (Conforms)