DATASHEET
Formulation
White or off-white lyophilize solid
Storage:
-20°C
Product Information:
YM-254890 is a novel Gαq/11 inhibitor,1 U46619-induced platelet aggregation is inhibited but phorbol ester- or ionophore-induced aggregation is not2 (IC50 = 0.1-0.2 μM)1. It blocks Pasteurella multocida toxin-mediated activation of Gαq.3 A highly useful new tool for studying Gαq/11-coupled receptor signaling and resulting cellular events.4
Description:
CAS Number: 568580-02-9<br></br>Chemical Name: Gq inhibitor<br></br>Molecular Weight: 960.10<br></br>Formula: C46H69N7O15<br></br>Solubility: DMSO (10 mg/ml)<br></br>Physical Properties: White or off-white lyophilize solid<br></br>Purity: 95% by HPLC, NMR (Conforms)