DATASHEET
Formulation
White or off-white solid
Storage:
-20°C
Product Information:
Potent pan-specific protein kinase inhibitor: PKA (Ki = 18 nM), PKC (Ki = 25 nM) PKG (Ki = 20 nM)1. Inhibits CaMK (Ki = 1.8 nM)2 and phosphorylase kinase (IC50 = 1.7 nM)3 as well as other kinases4. Induces apoptosis5. Cell permeable.
Description:
CAS Number: 99533-80-9<br></br>Chemical Name: Kinase inhibitor (pan-specific)<br></br>Molecular Weight: 467.49<br></br>Formula: C27H21N3O5<br></br>Solubility: DMSO (100 mg/ml)<br></br>Physical Properties: White or off-white solid<br></br>Purity: 98% by TLC, NMR (Conforms)