bs-83236C [Life Science]
K252A
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Formulation White or off-white solid

Storage: -20°C

Product Information:

Potent pan-specific protein kinase inhibitor: PKA (Ki = 18 nM), PKC (Ki = 25 nM) PKG (Ki = 20 nM)1. Inhibits CaMK (Ki = 1.8 nM)2 and phosphorylase kinase (IC50 = 1.7 nM)3 as well as other kinases4. Induces apoptosis5. Cell permeable.

Description:

CAS Number: 99533-80-9<br></br>Chemical Name: Kinase inhibitor (pan-specific)<br></br>Molecular Weight: 467.49<br></br>Formula: C27H21N3O5<br></br>Solubility: DMSO (100 mg/ml)<br></br>Physical Properties: White or off-white solid<br></br>Purity: 98% by TLC, NMR (Conforms)

Size: 5mg, 1mg

Applications: Life Science

For research use only. Not intended for diagnostic or therapeutic use.