DATASHEET
Formulation
Yellow solid
Storage:
RT
Product Information:
A potent and selective inhibitor of PARP1 and 2. EC50 = 20 nM1. Reduces ischemia reperfusion injury in a mouse model.2 Displays anti-inflammatory effects in a transient focal cerebral ischemia mouse model.3 Causes PARP1 independent, p21 dependent mitotic arrest.4
Description:
CAS Number: 344458-15-7<br></br>Chemical Name: PARP1,2 inhibitor<br></br>Molecular Weight: 331.81<br></br>Formula: C17H17N3O2<br></br>Solubility: DMSO (30mg/ml) Water (20 mg/ml)<br></br>Physical Properties: Yellow solid<br></br>Purity: 98% by HPLC NMR (Conforms)