DATASHEET
Formulation
Yellow solid
Storage:
-20°C
Product Information:
UH15-38 is a potent (IC50 = 20 nM) inhibitor of RIPK3 with excellent cellular activity. It blocked TNF-induced necroptosis in primary mouse embryonic fibroblasts (IC50 = 98 nM). UH15-38 selectively blocked influenza A-induced necroptosis over apoptosis in mouse alveolar epithelial cells, mouse embryonic fibroblasts, and human M29 cells at nanomolar levels. It attenuated influenza A-induced lung injury and lethality in vivo.
Description:
CAS Number: 2540881-21-6 (free base)<br></br>Chemical Name: RIP3K inhibitor<br></br>Molecular Weight: 514.45<br></br>Formula: C26H27N5O·2HCl<br></br>Solubility: DMSO (5 mg/ml) Water (>20 mg/ml)<br></br>Physical Properties: Yellow solid<br></br>Purity: >98% by HPLC NMR (Conforms)