DATASHEET
Formulation
Dark red to light brown solid
Storage:
-20°C
Product Information:
Potent and specific inhibitor of protein kinase C (PKC, IC50 = 50 nM).1 Inhibition of PKC is light dependent2 and is competitive with the diacylglycerol / phorbol ester binding site1. Calphostin C competes with the diacylglycerol / phorbol ester binding site in other proteins such as Munc13-1.3 Reverses oxycodone-induced tolerance to respiratory depression.4
Description:
CAS Number: 121263-19-2<br></br>Chemical Name: Protein Kinase C inhibitor<br></br>Molecular Weight: 790.77<br></br>Formula: C44H38O14<br></br>Solubility: DMSO (10 mg/ml)<br></br>Physical Properties: Dark red to light brown solid<br></br>Purity: 98% by HPLC NMR (Conforms)