bs-83812C [Life Science]
AT7519 HCl
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Formulation White solid

Storage: -20°C

Product Information:

AT7519 is a potent CDK inhibitor. Inhibits CDKs 1,2,4,5,6, and 9 (IC50s respectively: 210 nM, 47 nM, 100 nM, 13 nM, 170 nM, and <10 nM).1,2 Active in multiple human cancer cell lines.3-7 AT7519 has also been found to be a human RORγt agonist.8

Description:

CAS Number: 902135-91-5<br></br>Chemical Name: 4-[(2,6-Dichlorobenzoyl)amino]-N-piperidin-4-yl-1H-pyrazole-5-carboxamide hydrochloride<br></br>Molecular Weight: 418.7<br></br>Formula: C16H17Cl2N5O2·HCl<br></br>Solubility: DMSO (>25 mg/ml)<br></br>Physical Properties: White solid<br></br>Purity: >98% by HPLC NMR (Conforms)

Size: 5mg, 25mg

Applications: Life Science

For research use only. Not intended for diagnostic or therapeutic use.